Bicyclic Derivatives of the Potent Dual Aromatase–Steroid Sulfatase Inhibitor 2-Bromo-4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities
Paul M. Wood, L. W. Lawrence Woo, Jean-Robert Labrosse, Mark P. Thomas, Mary F. Mahon, Surinder K. Chander, Atul Purohit, Michael J. Reed, Barry V. L. PotterТом:
5
Рік:
2010
Мова:
english
Сторінки:
17
DOI:
10.1002/cmdc.201000203
Файл:
PDF, 697 KB
english, 2010