Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV inhibitor
Noriyasu Kato, Mitsuru Oka, Takayo Murase, Masahiro Yoshida, Masao Sakairi, Satoko Yamashita, Yoshika Yasuda, Aya Yoshikawa, Yuuji Hayashi, Mitsuhiro Makino, Motohiro Takeda, Yakufu Mirensha, Takuji KТом:
19
Рік:
2011
Мова:
english
Сторінки:
7
DOI:
10.1016/j.bmc.2011.09.043
Файл:
PDF, 535 KB
english, 2011