Identification of a Brain Penetrant PDE9A Inhibitor Utilizing Prospective Design and Chemical Enablement as a Rapid Lead Optimization Strategy
Verhoest, Patrick R., Proulx-Lafrance, Caroline, Corman, Michael, Chenard, Lois, Helal, Christopher J., Hou, Xinjun, Kleiman, Robin, Liu, Shenping, Marr, Eric, Menniti, Frank S., Schmidt, ChristopherТом:
52
Мова:
english
Журнал:
Journal of Medicinal Chemistry
DOI:
10.1021/jm9015334
Date:
December, 2009
Файл:
PDF, 3.28 MB
english, 2009