Discovery of selective, orally bioavailable, N -linked arylsulfonamide Na v 1.7 inhibitors with pain efficacy in mice
Roecker, Anthony J., Egbertson, Melissa, Jones, Kristen L.G., Gomez, Robert, Kraus, Richard L., Li, Yuxing, Koser, Amy Jo, Urban, Mark O., Klein, Rebecca, Clements, Michelle, Panigel, Jacqueline, DaleТом:
27
Мова:
english
Журнал:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2017.03.085
Date:
May, 2017
Файл:
PDF, 689 KB
english, 2017