Пожертвування 15 вересня 2024 – 1 жовтня 2024 Про збір коштів

Volume 10; Issue 9

Bioorganic & Medicinal Chemistry

Volume 10; Issue 9

1

QSAR Studies on Carbonic Anhydrase Inhibitors: A Case of Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides

Vijay K. Agrawal, Ruchi Sharma, Padmakar V. Khadikar

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 139 KB

english, 2002

2

Hydrazinocurcumin, a novel synthetic curcumin derivative, is a potent inhibitor of endothelial cell proliferation

Joong Sup Shim, Dong Hoon Kim, Hye Jin Jung, Jin Hee Kim, Dongyeol Lim, Seok-Ki Lee, Kyu-Won Kim, Jong Woong Ahn, Jong-Shin Yoo, Jung-Rae Rho, Jongheon Shin, Ho Jeong Kwon

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 213 KB

english, 2002

3

CYP3A4 Inhibitory Activity of New Bisalkaloids, Dipiperamides D and E, and Cognates from White Pepper

Sachiko Tsukamoto, Kyoko Tomise, Keiko Miyakawa, Bae-Cheon Cha, Takamasa Abe, Toshiyuki Hamada, Hiroshi Hirota, Tomihisa Ohta

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 147 KB

english, 2002

4

Adenine and Deazaadenine Nucleoside and Deoxynucleoside Analogues: Inhibition of Viral Replication of Sheep MVV (In Vitro Model for HIV) and Bovine BHV-1

Daniela Salvatori, Rosaria Volpini, Silvia Vincenzetti, Alberto Vita, Stefano Costanzi, Catia Lambertucci, Gloria Cristalli, Sauro Vittori

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 175 KB

english, 2002

5

Synthesis and Biological Activity of Novel Neuroprotective Diketopiperazines

K.R.C Prakash, Y Tang, Alan P Kozikowski, Judith L Flippen-Anderson, Susan M Knoblach, Alan I Faden

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 189 KB

english, 2002

6

Corrigendum to “metabolites of orally active NO-independent pyrazolopyridine stimulators of soluble guanylate cyclase”☆[Bioorg. Med. Chem. 10 (2002) 1711]

Alexander Straub, Jordi Benet-Buchholz, Rita Fröde, Armin Kern, Christian Kohlsdorfer, Peter Schmitt, Thomas Schwarz, Hans-Martin Siefert, Johannes-Peter Stasch

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 51 KB

english, 2002

7

Synthesis and Biological Evaluation of MAO-A Selective 1,4-Disubstituted-1,2,3,6-tetrahydropyridinyl Substrates

Philippe Bissel, Mark C Bigley, Kay Castagnoli, Neal Castagnoli Jr

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 230 KB

english, 2002

8

Molecular modeling of 3-arylisoquinoline antitumor agents active against A-549. A comparative molecular field analysis study

Won-Jea Cho, Eui-Ki Kim, Il Yeong Park, Eun Young Jeong, Tae Sung Kim, Thanh Nguyen Le, Dae-Duk Kim, Eung-Seok Lee

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 630 KB

english, 2002

9

Structure–activity relationships of benzylidene anabaseines in nicotinic acetylcholine receptors of cockroach nerve cords

Israt Sultana, Izumi Ikeda, Yoshihisa Ozoe

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 227 KB

english, 2002

10

Design, synthesis, and biological evaluation of a cephalosporin–monohydroguaiaretic acid prodrug activated by a monoclonal antibody–β-lactamase conjugate

Gholam Hossein Hakimelahi, Kak-Shan Shia, Manijeh Pasdar, Shahram Hakimelahi, Ali Khalafi-Nezhad, Mohammad N Soltani, Nai-Wen Mei, Hui-Ching Mei, Ali A Saboury, Mostafa Rezaei-Tavirani, Ali A Moosavi-

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 142 KB

english, 2002

11

Nucleosides and nucleotides. Part 214: thermal stability of triplexes containing 4′α-C-Aminoalkyl-2′-deoxynucleosides

Naoko Atsumi, Yoshihito Ueno, Makiko Kanazaki, Satoshi Shuto, Akira Matsuda

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 170 KB

english, 2002

12

In vitro antitumor activities of 2,6-di-[2-(Heteroaryl)vinyl]pyridines and pyridiniums

Vincenza Barresi, Daniele F Condorelli, Cosimo G Fortuna, Giuseppe Musumarra, Salvatore Scirè

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 131 KB

english, 2002

13

Novel potent substance P and neurokinin A receptor antagonists. Conception, synthesis and biological evaluation of indolizine derivatives

Régis Millet, Juozas Domarkas, Benoı̂t Rigo, Laurence Goossens, Jean-François Goossens, Raymond Houssin, Jean-Pierre Hénichart

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 181 KB

english, 2002

14

DNA damage and biological effects induced by photosensitization with new N1-unsubstituted furo[2,3-h]quinolin-2(1H)-ones

Cristina Marzano, Adriana Chilin, Franco Bordin, Francarosa Baccichetti, Adriano Guiotto

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 201 KB

english, 2002

15

Pyridazines. Part XXIX: synthesis and platelet aggregation inhibition activity of 5-substituted-6-phenyl-3(2H)-pyridazinones. Novel aspects of their biological actions

Eddy Sotelo, Nuria Fraiz, Matilde Yáñez, Vicente Terrades, Reyes Laguna, Ernesto Cano, Enrique Raviña

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 253 KB

english, 2002

16

Synthesis and cytotoxic evaluation of analogues of the marine pyridoacridine amphimedine

Christine Brahic, Francis Darro, Mirabelle Belloir, Jean Bastide, Robert Kiss, Evelyne Delfourne

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 195 KB

english, 2002

17

Sesquiterpene lactones as inhibitors of human neutrophil elastase

B Siedle, S Cisielski, R Murillo, B Löser, V Castro, C.A Klaas, O Hucke, A Labahn, M.F Melzig, I Merfort

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 219 KB

english, 2002

18

Synthesis and anti-inflammatory activity of phthalimide derivatives, designed as new thalidomide analogues

Lı́dia M Lima, Paulo Castro, Alexandre L Machado, Carlos Alberto M Fraga, Claire Lugnier, Vera Lúcia Gonçalves de Moraes, Eliezer J Barreiro

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 175 KB

english, 2002

19

Novel substrates for nitric oxide synthases

Ming Xian, Noriko Fujiwara, Zhong Wen, Tingwei Cai, Satoshi Kazuma, Adam J Janczuk, Xiaoping Tang, Vladislav V Telyatnikov, Yingxin Zhang, Xinchao Chen, Yasuhide Miyamoto, Naoyuki Taniguchi, Peng Geor

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 144 KB

english, 2002

20

Synthesis and characterization of a catalytic Antibody–HPMA copolymer-Conjugate as a tool for tumor selective prodrug activation

Ronit Satchi-Fainaro, Wolfgang Wrasidlo, Holger N Lode, Doron Shabat

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 227 KB

english, 2002

21

Novel furano analogues of duocarmycin C1 and C2: design, synthesis, and biological evaluation of seco-iso-Cyclopropylfurano[2,3-e]indoline (seco-iso-CFI) and seco-Cyclopropyltetrahydrofurano[2,3-f]quinoline (seco-CFQ) analogues

Tiffany T. Howard, Brian M. Lingerfelt, Bethany L. Purnell, Adrienne E. Scott, Carly A. Price, Heather M. Townes, LuAnne McNulty, Heather L. Handl, Kaitlin Summerville, Stephen J. Hudson, J.Phillip Bo

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 343 KB

english, 2002

22

QSAR studies on biological activity of piritrexim analogues against pc DHFR

Vijay K. Agrawal, Rashmi Sohgaura, Padmakar V. Khadikar

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 153 KB

english, 2002

23

Transport of the highly charged myo-inositol hexakisphosphate molecule across the red blood cell membrane: a phase transfer and biological study

Stéphane P Vincent, Jean-Marie Lehn, Jaime Lazarte, Claude Nicolau

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 223 KB

english, 2002

24

Cytotoxic T lymphocyte epitope analogues containing cis- or trans-4-aminocyclohexanecarboxylic acid residues

Mauro Marastoni, Martina Bazzaro, Fabiola Micheletti, Riccardo Gavioli, Roberto Tomatis

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 137 KB

english, 2002

25

Structural Studies on Bioactive Compounds. Part 36: Design, Synthesis and Biological Evaluation of Pyrimethamine-Based Antifolates Against Pneumocystis carinii

David C.M. Chan, Charles A. Laughton, Sherry F. Queener, Malcolm F.G. Stevens

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 311 KB

english, 2002

26

Synthesis of new 2,5-Disubstituted-1,3,4-thiadiazoles and preliminary evaluation of anticonvulsant and antimicrobial activities

Hatice N Dogan, Arzu Duran, Sevim Rollas, Göksel Sener, Meral K Uysal, Dumrul Gülen

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 136 KB

english, 2002

27

(Z)-1,4-Diamino-2-butene as a vector of boron, fluorine, or iodine for cancer therapy and imaging: synthesis and biological evaluation

Bénédicte Martin, Françoise Possémé, Caroline Le Barbier, François Carreaux, Bertrand Carboni, Nikolaus Seiler, Jacques-Philippe Moulinoux, Jean-Guy Delcros

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 185 KB

english, 2002

28

Superoxide dismutase mimetics: synthesis and structure–activity relationship study of MnTBAP analogues

Polivina Jolicia F Gauuan, Michael P Trova, Livia Gregor-Boros, Stephen B Bocckino, James D Crapo, Brian J Day

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 188 KB

english, 2002

29

Effects of 4,4-Dimethyl-5,8-dihydroxynaphtalene-1-one and 4,4-Dimethyl-5,8-dihydroxytetralone derivatives on tumor cell respiration

Ramiro Araya-Maturana, Tomás Delgado-Castro, Mario Gárate, Jorge Ferreira, Mario Pavani, Hernán Pessoa-Mahana, Bruce K Cassels

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 94 KB

english, 2002

30

QSAR study on competition binding of rodenticides (PATs) to H1 receptor in rat and guinea pig brain

Vijay K. Agrawal, Sanjay Karmarkar, Padmakar V. Khadikar

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 131 KB

english, 2002

31

Molecular docking and 3-D-QSAR studies on the possible antimalarial mechanism of artemisinin analogues

Feng Cheng, Jianhua Shen, Xiaomin Luo, Weiliang Zhu, Jiande Gu, Ruyun Ji, Hualiang Jiang, Kaixian Chen

Журнал:

Bioorganic & Medicinal Chemistry

Рік:

2002

Мова:

english

Файл:

PDF, 262 KB

english, 2002